The novel autophagy inhibitor ROC-325 augments the antileukemic activity of azacitidine

Leukemia. 2019 Dec;33(12):2971-2974. doi: 10.1038/s41375-019-0529-2. Epub 2019 Jul 29.
No abstract available

Publication types

  • Letter
  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Antimetabolites, Antineoplastic / pharmacology*
  • Autophagy / drug effects*
  • Azacitidine / pharmacology*
  • Cell Line, Tumor
  • Drug Synergism
  • Humans
  • Hydroxychloroquine / analogs & derivatives
  • Hydroxychloroquine / pharmacology
  • Mice
  • Xenograft Model Antitumor Assays

Substances

  • 1-(2-(2-((7-chloroquinolin-4-yl)amino)ethyl-methylamino)ethylamino)-4-methylthioxanthen-9-one
  • Antimetabolites, Antineoplastic
  • Hydroxychloroquine
  • Azacitidine