The comprehensive review contains the analysis of literature data concerning reactions of heterocyclization of aminoazoles and demonstrates the application of these types of transformations in diversity-oriented synthesis. The review is oriented to wide range of chemists working in the field of organic synthesis and both experimental and theoretical studies of nitrogen-containing heterocycles.
Keywords: aminoazole; click-chemistry; diversity-oriented synthesis; heterocycle; heterocyclization reaction; microwave-assisted organic synthesis; multicomponent reaction; ultrasonication.