Constrained peptides and biological targets

Bioorg Med Chem. 2018 Mar 15;26(6):1117. doi: 10.1016/j.bmc.2018.02.046.
No abstract available

Publication types

  • Editorial

MeSH terms

  • Cyclization
  • ErbB Receptors / antagonists & inhibitors
  • ErbB Receptors / metabolism
  • Humans
  • Peptides / chemical synthesis
  • Peptides / chemistry*
  • Peptides / metabolism
  • Phosphoprotein Phosphatases / chemistry
  • Phosphoprotein Phosphatases / metabolism
  • Receptors, Opioid, kappa / antagonists & inhibitors
  • Receptors, Opioid, kappa / metabolism
  • Structure-Activity Relationship

Substances

  • Peptides
  • Receptors, Opioid, kappa
  • EGFR protein, human
  • ErbB Receptors
  • Phosphoprotein Phosphatases