Dual blockade of the lipid kinase PIP4Ks and mitotic pathways leads to cancer-selective lethality

Nat Commun. 2017 Dec 19;8(1):2200. doi: 10.1038/s41467-017-02287-5.

Abstract

Achieving robust cancer-specific lethality is the ultimate clinical goal. Here, we identify a compound with dual-inhibitory properties, named a131, that selectively kills cancer cells, while protecting normal cells. Through an unbiased CETSA screen, we identify the PIP4K lipid kinases as the target of a131. Ablation of the PIP4Ks generates a phenocopy of the pharmacological effects of PIP4K inhibition by a131. Notably, PIP4Ks inhibition by a131 causes reversible growth arrest in normal cells by transcriptionally upregulating PIK3IP1, a suppressor of the PI3K/Akt/mTOR pathway. Strikingly, Ras activation overrides a131-induced PIK3IP1 upregulation and activates the PI3K/Akt/mTOR pathway. Consequently, Ras-transformed cells override a131-induced growth arrest and enter mitosis where a131's ability to de-cluster supernumerary centrosomes in cancer cells eliminates Ras-activated cells through mitotic catastrophe. Our discovery of drugs with a dual-inhibitory mechanism provides a unique pharmacological strategy against cancer and evidence of cross-activation between the Ras/Raf/MEK/ERK and PI3K/AKT/mTOR pathways via a Ras˧PIK3IP1˧PI3K signaling network.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acrylonitrile / analogs & derivatives*
  • Acrylonitrile / pharmacology
  • Acrylonitrile / therapeutic use
  • Animals
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Cell Survival / drug effects
  • Female
  • Humans
  • Indoles / pharmacology*
  • Indoles / therapeutic use
  • Intracellular Signaling Peptides and Proteins
  • Isoquinolines / pharmacology*
  • Isoquinolines / therapeutic use
  • Membrane Proteins / metabolism*
  • Mice
  • Mice, Inbred BALB C
  • Mice, Nude
  • Mitosis / drug effects*
  • Neoplasms / drug therapy*
  • Phosphotransferases (Alcohol Group Acceptor) / antagonists & inhibitors*
  • Protein Kinase Inhibitors / pharmacology*
  • Protein Kinase Inhibitors / therapeutic use
  • Signal Transduction / drug effects*
  • Xenograft Model Antitumor Assays
  • ras Proteins / metabolism

Substances

  • A131 compound
  • Indoles
  • Intracellular Signaling Peptides and Proteins
  • Isoquinolines
  • Membrane Proteins
  • PIK3IP1 protein, human
  • Protein Kinase Inhibitors
  • Phosphotransferases (Alcohol Group Acceptor)
  • ras Proteins
  • Acrylonitrile