Drugging the undruggable: targeting challenging E3 ligases for personalized medicine

Future Med Chem. 2017 Mar;9(4):347-350. doi: 10.4155/fmc-2017-0009. Epub 2017 Mar 6.
No abstract available

Keywords: E3 ligases; personalized medicine; protein–protein interactions; undruggable targets.

Publication types

  • Editorial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Drug Discovery
  • Enzyme Inhibitors / chemistry
  • Enzyme Inhibitors / pharmacology*
  • Humans
  • Ligands
  • Precision Medicine*
  • Ubiquitin-Protein Ligases / antagonists & inhibitors*
  • Ubiquitin-Protein Ligases / metabolism

Substances

  • Enzyme Inhibitors
  • Ligands
  • Ubiquitin-Protein Ligases