Are fluoxetine's effects due to sigma-1 receptor agonism?

Pharmacol Res. 2016 Nov;113(Pt A):707-708. doi: 10.1016/j.phrs.2016.05.031. Epub 2016 Jun 2.
No abstract available

Publication types

  • Letter

MeSH terms

  • Animals
  • Antidepressive Agents, Second-Generation / metabolism
  • Antidepressive Agents, Second-Generation / pharmacology*
  • Fluoxetine / metabolism
  • Fluoxetine / pharmacology*
  • Humans
  • Receptors, sigma / agonists*
  • Receptors, sigma / metabolism
  • Sigma-1 Receptor

Substances

  • Antidepressive Agents, Second-Generation
  • Receptors, sigma
  • Fluoxetine