Regioselective synthesis of 2H-indazoles through Ga/Al- and Al-mediated direct alkylation reactions of indazoles

Org Biomol Chem. 2015 Dec 14;13(46):11376-81. doi: 10.1039/c5ob01747e.

Abstract

A procedure has been developed for the regioselective, high yielding synthesis of 2H-indazoles that involves direct alkylation of indazoles with various allyl and benzyl bromides, and α-bromocarbonyl compounds.

Publication types

  • Research Support, Non-U.S. Gov't