Abstract
A synergistic dual-targeting molecular self-assembly hydrogel was designed with estrone (Et) and Arg-Gly-Asp (RGD) peptide. Confocal imaging in vitro and real-time visualization in vivo researches were carried out to evidence enhanced targeted delivery and anticancer effect of Taxol.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Animals
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Antineoplastic Agents, Phytogenic / administration & dosage*
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Antineoplastic Agents, Phytogenic / chemistry
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Antineoplastic Agents, Phytogenic / pharmacokinetics
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Breast Neoplasms / metabolism
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Cell Survival / drug effects
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Coloring Agents / chemistry
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Drug Carriers* / administration & dosage
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Drug Carriers* / chemistry
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Drug Carriers* / pharmacokinetics
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Estrone* / administration & dosage
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Estrone* / chemistry
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Estrone* / pharmacokinetics
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Female
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Humans
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Hydrogels* / administration & dosage
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Hydrogels* / chemistry
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Hydrogels* / pharmacokinetics
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Indocyanine Green / chemistry
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MCF-7 Cells
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Mice, Nude
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Oligopeptides* / administration & dosage
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Oligopeptides* / chemistry
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Oligopeptides* / pharmacokinetics
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Paclitaxel / administration & dosage*
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Paclitaxel / chemistry
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Paclitaxel / pharmacokinetics
Substances
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Antineoplastic Agents, Phytogenic
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Coloring Agents
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Drug Carriers
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Hydrogels
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Oligopeptides
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Estrone
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arginyl-glycyl-aspartic acid
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Indocyanine Green
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Paclitaxel