Sequential one-pot access to molecular diversity through aniline aqueous borylation

J Org Chem. 2014 Nov 7;79(21):10568-80. doi: 10.1021/jo501665e. Epub 2014 Oct 9.

Abstract

On the basis of our recently reported aniline aqueous borylation, molecular diversity was achieved in a one-pot process by combining other reactions such as esterification, Suzuki-Miyaura coupling, hydrogenolysis, or Petasis borono-Mannich.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aniline Compounds / chemistry*
  • Benzoxazoles / chemical synthesis*
  • Benzoxazoles / chemistry
  • Boron Compounds / chemical synthesis*
  • Boron Compounds / chemistry
  • Boronic Acids / chemical synthesis*
  • Boronic Acids / chemistry
  • Catalysis
  • Molecular Structure
  • Palladium / chemistry

Substances

  • 2-oxo-2,3-dihydrobenzo(d)oxazol-6-ylboronic acid
  • Aniline Compounds
  • Benzoxazoles
  • Boron Compounds
  • Boronic Acids
  • Palladium
  • aniline