Antimalarial tropones and their Plasmodium falciparum glyoxalase I (pfGLOI) inhibitory activity

J Antibiot (Tokyo). 2014 Jul;67(7):545-7. doi: 10.1038/ja.2014.28. Epub 2014 Apr 9.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antimalarials / chemistry*
  • Enzyme Inhibitors / chemistry
  • Enzyme Inhibitors / pharmacology
  • Lactoylglutathione Lyase / antagonists & inhibitors*
  • Penicillium / chemistry
  • Plasmodium falciparum / drug effects*
  • Tropolone / analogs & derivatives*
  • Tropolone / chemistry
  • Tropolone / pharmacology

Substances

  • Antimalarials
  • Enzyme Inhibitors
  • Tropolone
  • tropone
  • Lactoylglutathione Lyase