A new development in DNA repair modulation: discovery of a BLM helicase inhibitor

Cell Cycle. 2013 Mar 1;12(5):713-4. doi: 10.4161/cc.23953. Epub 2013 Feb 19.
No abstract available

Keywords: Bloom's syndrome; DNA repair; RecQ; anticancer therapy; helicase; high-throughput screening; inhibitor; molecular probes; small molecules; synthetic lethality.

Publication types

  • Editorial

MeSH terms

  • DNA Helicases / antagonists & inhibitors*
  • DNA Helicases / chemistry
  • DNA Helicases / metabolism
  • DNA Repair / drug effects*
  • Enzyme Inhibitors / pharmacology*
  • Humans
  • Poly(ADP-ribose) Polymerase Inhibitors
  • Poly(ADP-ribose) Polymerases / metabolism
  • RecQ Helicases / antagonists & inhibitors*
  • RecQ Helicases / chemistry
  • RecQ Helicases / metabolism
  • Small Molecule Libraries / pharmacology

Substances

  • Enzyme Inhibitors
  • Poly(ADP-ribose) Polymerase Inhibitors
  • Small Molecule Libraries
  • Poly(ADP-ribose) Polymerases
  • Bloom syndrome protein
  • DNA Helicases
  • RecQ Helicases