Conformational selection versus induced fit in kinases: the case of PI3K-γ

Angew Chem Int Ed Engl. 2012 Jan 16;51(3):642-6. doi: 10.1002/anie.201103264. Epub 2011 Dec 1.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoproteins / chemistry
  • Apoproteins / metabolism
  • Binding Sites
  • Humans
  • Ligands
  • Molecular Dynamics Simulation
  • Phosphatidylinositol 3-Kinases / chemistry*
  • Phosphatidylinositol 3-Kinases / metabolism
  • Protein Binding
  • Protein Conformation

Substances

  • Apoproteins
  • Ligands
  • Phosphatidylinositol 3-Kinases
  • PIK3R3 protein, human