Specific targeting of hypoxic tumor tissue with nitroimidazole-peptide conjugates

ChemMedChem. 2012 Jan 2;7(1):57-61. doi: 10.1002/cmdc.201100401. Epub 2011 Sep 29.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Cell-Penetrating Peptides / chemistry*
  • Drug Delivery Systems*
  • Hypoxia / drug therapy*
  • Metronidazole / administration & dosage*
  • Metronidazole / chemistry
  • Metronidazole / pharmacokinetics
  • Molecular Sequence Data
  • Neoplasms / drug therapy*
  • Radiation-Sensitizing Agents / administration & dosage*
  • Radiation-Sensitizing Agents / chemistry
  • Radiation-Sensitizing Agents / pharmacokinetics
  • Rats
  • Rats, Wistar

Substances

  • Cell-Penetrating Peptides
  • Radiation-Sensitizing Agents
  • Metronidazole