Variation in binding affinity of the novel anxiolytic XBD173 for the 18 kDa translocator protein in human brain

Synapse. 2011 Mar;65(3):257-9. doi: 10.1002/syn.20884.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Anxiety Agents / metabolism*
  • Brain / metabolism*
  • Humans
  • Protein Binding
  • Purines / metabolism*
  • Receptors, GABA / metabolism*

Substances

  • Anti-Anxiety Agents
  • N-benzyl-N-ethyl-2-(7,8-dihydro-7-methyl-8-oxo-2-phenyl-9H-purin-9-yl)acetamide
  • Purines
  • Receptors, GABA
  • TSPO protein, human