Small-molecule inhibitors of the ERK signaling pathway: Towards novel anticancer therapeutics

ChemMedChem. 2011 Jan 3;6(1):38-48. doi: 10.1002/cmdc.201000354.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Antineoplastic Agents / metabolism
  • Antineoplastic Agents / pharmacology*
  • Cell Line, Tumor
  • Enzyme Inhibitors / metabolism
  • Enzyme Inhibitors / pharmacology*
  • Extracellular Signal-Regulated MAP Kinases / antagonists & inhibitors*
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • Humans
  • MAP Kinase Signaling System / drug effects
  • Mice
  • Neoplasms / drug therapy
  • Protein Binding / drug effects
  • Quantitative Structure-Activity Relationship
  • Signal Transduction / drug effects
  • Small Molecule Libraries / metabolism
  • Small Molecule Libraries / pharmacology*
  • raf Kinases / antagonists & inhibitors*
  • raf Kinases / metabolism

Substances

  • Antineoplastic Agents
  • Enzyme Inhibitors
  • Small Molecule Libraries
  • raf Kinases
  • Extracellular Signal-Regulated MAP Kinases