Preparation of benzolactams by Pd(II)-catalyzed carbonylation of N-unprotected arylethylamines

Chem Commun (Camb). 2011 Jan 21;47(3):1054-6. doi: 10.1039/c0cc03478a. Epub 2010 Nov 15.

Abstract

An unprecedented NH(2)-directed Pd(II)-catalytic carbonylation of quaternary aromatic α-amino esters to yield 6-membered benzolactams has been developed. The reaction shows a strong bias to 6-membered lactams over 5-membered ones. The steric hindrance around the amino group seems to be pivotal for the success of the process.