In silico characterization of ligand binding modes in the human histamine H4 receptor and their impact on receptor activation

Chembiochem. 2010 Sep 3;11(13):1850-5. doi: 10.1002/cbic.201000180.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Drug Inverse Agonism
  • Humans
  • Hydrogen Bonding
  • Ligands*
  • Molecular Dynamics Simulation
  • Protein Binding
  • Protein Structure, Tertiary
  • Pyrimidines / chemistry
  • Receptors, G-Protein-Coupled / antagonists & inhibitors
  • Receptors, G-Protein-Coupled / metabolism*
  • Receptors, Histamine / metabolism*
  • Receptors, Histamine H4

Substances

  • HRH4 protein, human
  • Ligands
  • Pyrimidines
  • Receptors, G-Protein-Coupled
  • Receptors, Histamine
  • Receptors, Histamine H4