Promising lead compounds for novel antiprotozoals

J Antibiot (Tokyo). 2010 Jul;63(7):381-4. doi: 10.1038/ja.2010.50. Epub 2010 May 26.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Bacterial Agents / chemistry
  • Anti-Bacterial Agents / pharmacology
  • Antibiotics, Antineoplastic / chemistry
  • Antibiotics, Antineoplastic / pharmacology
  • Antimalarials / chemistry
  • Antimalarials / pharmacology
  • Antiprotozoal Agents / chemistry*
  • Antiprotozoal Agents / pharmacology*
  • Cell Line, Tumor
  • Drug Screening Assays, Antitumor
  • Humans
  • In Vitro Techniques
  • Lysine / analogs & derivatives
  • Lysine / chemistry
  • Lysine / pharmacology
  • Malaria / drug therapy
  • Pactamycin / chemistry
  • Pactamycin / pharmacology
  • Parasitic Sensitivity Tests
  • Plasmodium falciparum / drug effects
  • Structure-Activity Relationship
  • Trypanocidal Agents / chemistry
  • Trypanocidal Agents / pharmacology
  • Trypanosoma brucei brucei / drug effects
  • Trypanosomiasis, African / drug therapy

Substances

  • Anti-Bacterial Agents
  • Antibiotics, Antineoplastic
  • Antimalarials
  • Antiprotozoal Agents
  • Trypanocidal Agents
  • beta-lysylmethanediamine
  • Pactamycin
  • Lysine