PND-1186 FAK inhibitor selectively promotes tumor cell apoptosis in three-dimensional environments

Cancer Biol Ther. 2010 May 15;9(10):791-3. doi: 10.4161/cbt.11729. Epub 2010 May 8.
No abstract available

Publication types

  • Comment

MeSH terms

  • Aminopyridines / pharmacology*
  • Animals
  • Antineoplastic Agents / pharmacology*
  • Apoptosis / drug effects*
  • Carrier Proteins / metabolism
  • Cell Survival / drug effects
  • Focal Adhesion Protein-Tyrosine Kinases / antagonists & inhibitors*
  • Mice
  • Protein Binding / drug effects
  • Protein Kinase Inhibitors / pharmacology*
  • Signal Transduction / drug effects
  • Spheroids, Cellular / drug effects
  • Tumor Cells, Cultured

Substances

  • Aminopyridines
  • Antineoplastic Agents
  • Carrier Proteins
  • PND 1186
  • Protein Kinase Inhibitors
  • Focal Adhesion Protein-Tyrosine Kinases