Antipain Y, a new antipain analog that inhibits neurotransmitter release from rat dorsal root ganglion neurons

J Antibiot (Tokyo). 2010 Jan;63(1):41-4. doi: 10.1038/ja.2009.109. Epub 2009 Nov 13.
No abstract available

MeSH terms

  • Animals
  • Antipain / chemistry*
  • Antipain / pharmacology*
  • Calcium / metabolism
  • Ganglia, Spinal / drug effects*
  • Mass Spectrometry
  • Molecular Structure
  • Neurons / drug effects*
  • Neurotransmitter Agents / antagonists & inhibitors*
  • Protease Inhibitors / chemistry*
  • Protease Inhibitors / pharmacology*
  • Rats
  • Substance P / antagonists & inhibitors*
  • Synaptic Transmission / drug effects
  • Trypsin / metabolism
  • Tryptases / antagonists & inhibitors

Substances

  • Neurotransmitter Agents
  • Protease Inhibitors
  • Substance P
  • Antipain
  • Trypsin
  • Tryptases
  • Calcium