Rational design of peptidomimetics for class B GPCRs: potent non-peptide GLP-1 receptor agonists

Adv Exp Med Biol. 2009:611:125-6. doi: 10.1007/978-0-387-73657-0_55.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Crystallography, X-Ray
  • Drug Design*
  • Glucagon-Like Peptide-1 Receptor
  • Models, Molecular
  • Molecular Mimicry*
  • Nuclear Magnetic Resonance, Biomolecular
  • Peptides / chemistry*
  • Peptides / pharmacology*
  • Protein Conformation
  • Receptors, Glucagon / agonists*

Substances

  • Glucagon-Like Peptide-1 Receptor
  • Peptides
  • Receptors, Glucagon