Cytochrome P450 metabolism and inhibition: analysis for drug discovery

Prog Med Chem. 2009:47:239-63. doi: 10.1016/S0079-6468(08)00206-3.
No abstract available

Publication types

  • Review

MeSH terms

  • Cytochrome P-450 Enzyme Inhibitors
  • Cytochrome P-450 Enzyme System / metabolism*
  • Drug Discovery / methods*
  • Enzyme Inhibitors / pharmacology*
  • Humans
  • Liver / enzymology
  • Pharmaceutical Preparations / metabolism
  • Structure-Activity Relationship
  • Substrate Specificity

Substances

  • Cytochrome P-450 Enzyme Inhibitors
  • Enzyme Inhibitors
  • Pharmaceutical Preparations
  • Cytochrome P-450 Enzyme System