Target flexibility: an emerging consideration in drug discovery and design

J Med Chem. 2008 Oct 23;51(20):6237-55. doi: 10.1021/jm800562d. Epub 2008 Sep 12.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Computer Simulation
  • Crystallography, X-Ray
  • Drug Design*
  • Drug Evaluation, Preclinical
  • Humans
  • Nuclear Magnetic Resonance, Biomolecular
  • Pharmaceutical Preparations / chemistry
  • Proteins / chemistry
  • Proteins / metabolism

Substances

  • Pharmaceutical Preparations
  • Proteins