A strategy to discover inhibitors of O-linked glycosylation

J Am Chem Soc. 2008 Jan 16;130(2):440-1. doi: 10.1021/ja078125s. Epub 2007 Dec 20.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Drug Evaluation, Preclinical
  • Endopeptidase K / chemistry*
  • Enzyme Inhibitors / chemistry*
  • Enzyme Inhibitors / pharmacology
  • Glycosylation / drug effects
  • Glycosyltransferases / antagonists & inhibitors*
  • Humans
  • Molecular Sequence Data
  • Peptides / chemistry
  • Proteins / chemistry
  • Proteins / metabolism*

Substances

  • Enzyme Inhibitors
  • Peptides
  • Proteins
  • Glycosyltransferases
  • Endopeptidase K