Pharmacokinetics of eprinomectin in plasma and milk following subcutaneous administration to lactating dairy cattle

Vet Res Commun. 2006 Apr;30(3):263-70. doi: 10.1007/s11259-006-3230-7.

Abstract

Eprinomectin is only available as a topically applied anthelmintic for dairy cattle. To determine whether eprinomectin can be applied as an injectable formulation in dairy cattle, a novel injectable formulation was developed and was subcutaneously delivered to four lactating dairy cattle at a dose rate of 0.2 mg/ kg. Plasma and milk samples were collected. The concentrations of eprinomectin in all samples were determined by HPLC. The peak plasma concentration (C(max))of 44.0+/-24.2 ng/ml occurred 39+/-19.3 h after subcutaneous administration, equivalent to the C(max) (43.76+/-18.23 ng/ml) previously reported for dairy cattle after a pour-on administration of 0.5 mg/kg eprinomectin. The area under the plasma concentration-time curve (AUC) after subcutaneous administration was 7354+/-1861 (ng h)/ml, higher than that obtained after pour-on delivery (5737.68+/-412.80 (ng h)/ml). The mean residence time (MRT) of the drug in plasma was 211+/-55.2 h. Eprinomectin was detected in the milk at the second sampling time. The concentration of drug in milk was parallel to that in plasma, with a milk to plasma ratio of 0.16+/-0.01. The highest detected concentration of eprinomectin in milk was 9.0 ng/ml, below the maximum residue limit (MRL) of eprinomectin in milk established by the Joint FAO/WHO Expert Committee on Food Additives in 2000. The amount of eprinomectin recovered in the milk during this trial was 0.39%+/-0.08% of the total administered dose. This study demonstrates that subcutaneous administration of eprinomectin led to higher bioavailability and a lower dose than a pour-on application, and that an injectable formulation of eprinomectin may be applied in dairy cattle with a zero withdrawal period.

Publication types

  • Clinical Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anthelmintics / administration & dosage
  • Anthelmintics / analysis
  • Anthelmintics / blood
  • Anthelmintics / pharmacokinetics*
  • Area Under Curve
  • Cattle
  • Female
  • Half-Life
  • Injections, Subcutaneous
  • Ivermectin / administration & dosage
  • Ivermectin / analogs & derivatives*
  • Ivermectin / analysis
  • Ivermectin / blood
  • Ivermectin / pharmacokinetics
  • Lactation
  • Milk / chemistry*

Substances

  • Anthelmintics
  • Ivermectin
  • eprinomectin