Discovering drugs through biological transformation: role of pharmacologically active metabolites in drug discovery

J Med Chem. 2004 Aug 26;47(18):4339-51. doi: 10.1021/jm040066v.
No abstract available

Publication types

  • Review

MeSH terms

  • Biotransformation*
  • Cytochrome P-450 Enzyme System / metabolism
  • Drug Design*
  • Drug Evaluation, Preclinical / methods
  • Pharmaceutical Preparations / chemistry
  • Pharmaceutical Preparations / isolation & purification
  • Pharmaceutical Preparations / metabolism

Substances

  • Pharmaceutical Preparations
  • Cytochrome P-450 Enzyme System