Structure-based design, synthesis, and in vitro evaluation of nonpeptidic neprilysin inhibitors

Chembiochem. 2004 Jul 5;5(7):996-1000. doi: 10.1002/cbic.200400005.
No abstract available

Publication types

  • Evaluation Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Drug Design*
  • Drug Evaluation
  • Enzyme Inhibitors / chemical synthesis*
  • Enzyme Inhibitors / chemistry
  • Enzyme Inhibitors / pharmacology*
  • Imidazoles / chemistry
  • In Vitro Techniques
  • Models, Molecular
  • Neprilysin / antagonists & inhibitors*
  • Structure-Activity Relationship

Substances

  • Enzyme Inhibitors
  • Imidazoles
  • Neprilysin