Effects of the administration of spiramycin and tiamulin on in vivo complex formation and hepatic cytochrome P4503A (CYP3A)-dependent monooxygenases in rabbits

Vet Res Commun. 2003 Sep:27 Suppl 1:377-9. doi: 10.1023/b:verc.0000014184.56266.1a.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Aryl Hydrocarbon Hydroxylases / drug effects
  • Aryl Hydrocarbon Hydroxylases / genetics
  • Aryl Hydrocarbon Hydroxylases / metabolism*
  • Cytochrome P-450 CYP3A
  • Diterpenes / pharmacology*
  • Gene Expression Regulation, Enzymologic / drug effects
  • Liver / drug effects
  • Liver / enzymology*
  • Oxidoreductases, N-Demethylating / drug effects
  • Oxidoreductases, N-Demethylating / genetics
  • Oxidoreductases, N-Demethylating / metabolism*
  • Rabbits
  • Spiramycin / pharmacology*

Substances

  • Diterpenes
  • Spiramycin
  • tiamulin
  • Aryl Hydrocarbon Hydroxylases
  • Cytochrome P-450 CYP3A
  • Oxidoreductases, N-Demethylating