Mucoadhesive buccal patches of miconazole nitrate: in vitro/in vivo performance and effect of ageing

Int J Pharm. 2003 Oct 2;264(1-2):1-14. doi: 10.1016/s0378-5173(03)00371-5.

Abstract

Mucoadhesive patches containing 10mg miconazole nitrate were evaluated. The patches were prepared with ionic polymers, sodium carboxymethyl cellulose (SCMC) and chitosan, or non-ionic polymers, polyvinyl alcohol (PVA), hydroxyethyl cellulose (HEC) and hydroxypropylmethyl cellulose (HPMC). Convenient bioadhesion, acceptable elasticity, swelling and surface pH were obtained. Patches exhibited sustained release over more than 5h and the addition of polyvinyl pyrrolidone (PVP) generally enhanced the release rate. Optimum release behaviour was shown with patches containing 10% w/v PVA and 5% w/v PVP. Study of the in vivo release from this formulation revealed uniform and effective salivary levels with adequate comfort and compliance during at least 6h. On the contrary, in vivo release of the commercial oral gel product resulted in a burst and transient release of miconazole, which diminished sharply after the first hour of application. Storage of these patches for 6 months did not affect the elastic properties, however, enhanced release rates were observed due to marked changes in the crystal habit of the drug.

Publication types

  • Comparative Study

MeSH terms

  • Adhesiveness
  • Adjuvants, Pharmaceutic / chemistry
  • Administration, Buccal
  • Administration, Oral
  • Adult
  • Antifungal Agents / administration & dosage
  • Antifungal Agents / chemistry
  • Antifungal Agents / pharmacokinetics*
  • Carboxymethylcellulose Sodium / chemistry
  • Cellulose / analogs & derivatives*
  • Cellulose / chemistry
  • Chemistry, Pharmaceutical
  • Chitin / analogs & derivatives*
  • Chitin / chemistry
  • Chitosan
  • Cross-Over Studies
  • Delayed-Action Preparations
  • Drug Stability
  • Female
  • Humans
  • Hypromellose Derivatives
  • In Vitro Techniques
  • Male
  • Methylcellulose / analogs & derivatives
  • Methylcellulose / chemistry
  • Miconazole / administration & dosage
  • Miconazole / chemistry
  • Miconazole / pharmacokinetics*
  • Middle Aged
  • Mouth Mucosa / metabolism*
  • Polyvinyl Alcohol / chemistry
  • Time Factors

Substances

  • Adjuvants, Pharmaceutic
  • Antifungal Agents
  • Delayed-Action Preparations
  • Chitin
  • Hypromellose Derivatives
  • Miconazole
  • Polyvinyl Alcohol
  • Cellulose
  • hydroxyethylcellulose
  • Methylcellulose
  • Chitosan
  • Carboxymethylcellulose Sodium