"Inactive" excipients such as Cremophor can affect in vivo drug disposition

Clin Pharmacol Ther. 2003 May;73(5):394-6. doi: 10.1016/s0009-9236(03)00010-9.
No abstract available

Publication types

  • Comment

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / antagonists & inhibitors
  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / metabolism
  • Cardiotonic Agents / pharmacokinetics
  • Digoxin / pharmacokinetics
  • Excipients*
  • Humans
  • Pharmaceutical Preparations / metabolism*
  • Pharmacokinetics
  • Polyethylene Glycols*

Substances

  • ATP Binding Cassette Transporter, Subfamily B, Member 1
  • Cardiotonic Agents
  • Excipients
  • Pharmaceutical Preparations
  • cremophor
  • Polyethylene Glycols
  • Digoxin