Stereospecific synthesis of azetidine-cis-2,3-dicarboxylic acid

Yasushi Arakawa; Tomoaki Murakami; Yukimi Arakawa; Shigeyuki Yoshifuji

doi:10.1248/cpb.51.96

Stereospecific synthesis of azetidine-cis-2,3-dicarboxylic acid

Chem Pharm Bull (Tokyo). 2003 Jan;51(1):96-7. doi: 10.1248/cpb.51.96.

Authors

Yasushi Arakawa¹, Tomoaki Murakami, Yukimi Arakawa, Shigeyuki Yoshifuji

Affiliation

¹ Faculty of Pharmaceutical Sciences, Hokuriku University, Kanazawa, Japan. ya-arakawa@hokuriku-u.ac.jp

PMID: 12520137
DOI: 10.1248/cpb.51.96

Abstract

Electrocyclic reaction product of 1-(methoxycarbonyl)-1,2-dihydropyridine was stereospecifically converted by RuO(4) oxidation into azetidine-cis-2,3-dicarboxylic acid.

MeSH terms

Azetidines / chemical synthesis*
Dicarboxylic Acids / chemical synthesis*
Stereoisomerism

Substances

Azetidines
Dicarboxylic Acids