Natural product derived receptor tyrosine kinase inhibitors: identification of IGF1R, Tie-2, and VEGFR-3 inhibitors

Angew Chem Int Ed Engl. 2002 Apr 2;41(7):1174-8. doi: 10.1002/1521-3773(20020402)41:7<1174::aid-anie1174>3.0.co;2-v.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Amino Acid Sequence
  • Angiogenesis Inhibitors / chemistry*
  • Angiogenesis Inhibitors / pharmacology
  • Combinatorial Chemistry Techniques
  • Diterpenes / chemistry*
  • Diterpenes / pharmacology
  • Molecular Sequence Data
  • Neovascularization, Pathologic / drug therapy
  • Quinones / chemistry*
  • Quinones / pharmacology
  • Receptor Protein-Tyrosine Kinases / antagonists & inhibitors*
  • Receptor Protein-Tyrosine Kinases / genetics
  • Receptor, IGF Type 1 / antagonists & inhibitors*
  • Receptor, IGF Type 1 / genetics
  • Receptor, TIE-2
  • Sequence Alignment
  • Vascular Endothelial Growth Factor Receptor-3 / antagonists & inhibitors*
  • Vascular Endothelial Growth Factor Receptor-3 / genetics

Substances

  • Angiogenesis Inhibitors
  • Diterpenes
  • Quinones
  • Receptor Protein-Tyrosine Kinases
  • Receptor, IGF Type 1
  • Receptor, TIE-2
  • Vascular Endothelial Growth Factor Receptor-3