Amyloid-lowering isocoumarins are not direct inhibitors of gamma-secretase

Nat Cell Biol. 2002 May;4(5):E110-1; author reply E111-2. doi: 10.1038/ncb0502-e110b.
No abstract available

Publication types

  • Comment
  • Letter

MeSH terms

  • Amyloid Precursor Protein Secretases
  • Amyloid beta-Peptides / metabolism*
  • Amyloid beta-Protein Precursor / genetics
  • Amyloid beta-Protein Precursor / metabolism
  • Animals
  • Aspartic Acid Endopeptidases / antagonists & inhibitors
  • Aspartic Acid Endopeptidases / metabolism
  • Cell Line
  • Coumarins / chemistry
  • Coumarins / metabolism*
  • Endopeptidases / metabolism*
  • Enzyme Inhibitors / metabolism*
  • Humans

Substances

  • Amyloid beta-Peptides
  • Amyloid beta-Protein Precursor
  • Coumarins
  • Enzyme Inhibitors
  • Amyloid Precursor Protein Secretases
  • Endopeptidases
  • Aspartic Acid Endopeptidases
  • BACE1 protein, human