de Kock C - Search Results

1

Syntheses and in Vitro Antiplasmodial Activity of Aminoalkylated Chalcones and Analogues.

Wilhelm A, Kendrekar P, Noreljaleel AE, Abay ET, Bonnet SL, Wiesner L, de Kock C, Swart KJ, van der Westhuizen JH. Wilhelm A, et al. Among authors: de kock c. J Nat Prod. 2015 Aug 28;78(8):1848-58. doi: 10.1021/acs.jnatprod.5b00114. Epub 2015 Aug 3. J Nat Prod. 2015. PMID: 26235033

2

Cyclopalladated organosilane-tethered thiosemicarbazones: novel strategies for improving antiplasmodial activity.

Adams M, Barnard L, de Kock C, Smith PJ, Wiesner L, Chibale K, Smith GS. Adams M, et al. Among authors: de kock c. Dalton Trans. 2016 Apr 7;45(13):5514-20. doi: 10.1039/c5dt04918k. Epub 2016 Feb 25. Dalton Trans. 2016. PMID: 26911403

3

Improved antiparasitic activity by incorporation of organosilane entities into half-sandwich ruthenium(II) and rhodium(III) thiosemicarbazone complexes.

Adams M, de Kock C, Smith PJ, Land KM, Liu N, Hopper M, Hsiao A, Burgoyne AR, Stringer T, Meyer M, Wiesner L, Chibale K, Smith GS. Adams M, et al. Among authors: de kock c. Dalton Trans. 2015 Feb 7;44(5):2456-68. doi: 10.1039/c4dt03234a. Dalton Trans. 2015. PMID: 25559246

4

Design, synthesis, and In vitro antituberculosis activity of 2(5H)-Furanone derivatives.

Ngwane AH, Panayides JL, Chouteau F, Macingwana L, Viljoen A, Baker B, Madikane E, de Kock C, Wiesner L, Chibale K, Parkinson CJ, Mmutlane EM, van Helden P, Wiid I. Ngwane AH, et al. Among authors: de kock c. IUBMB Life. 2016 Aug;68(8):612-20. doi: 10.1002/iub.1526. Epub 2016 Jun 27. IUBMB Life. 2016. PMID: 27346745 Free article.

5

2,4-Diaminothienopyrimidines as orally active antimalarial agents.

González Cabrera D, Le Manach C, Douelle F, Younis Y, Feng TS, Paquet T, Nchinda AT, Street LJ, Taylor D, de Kock C, Wiesner L, Duffy S, White KL, Zabiulla KM, Sambandan Y, Bashyam S, Waterson D, Witty MJ, Charman SA, Avery VM, Wittlin S, Chibale K. González Cabrera D, et al. Among authors: de kock c. J Med Chem. 2014 Feb 13;57(3):1014-22. doi: 10.1021/jm401760c. Epub 2014 Jan 28. J Med Chem. 2014. PMID: 24446664

6

Oral lipid-based nanoformulation of tafenoquine enhanced bioavailability and blood stage antimalarial efficacy and led to a reduction in human red blood cell loss in mice.

Melariri P, Kalombo L, Nkuna P, Dube A, Hayeshi R, Ogutu B, Gibhard L, deKock C, Smith P, Wiesner L, Swai H. Melariri P, et al. Int J Nanomedicine. 2015 Feb 20;10:1493-503. doi: 10.2147/IJN.S76317. eCollection 2015. Int J Nanomedicine. 2015. PMID: 25759576 Free PMC article.

7

Design, Synthesis, and Evaluation of Novel Ferroquine and Phenylequine Analogues as Potential Antiplasmodial Agents.

Jacobs L, de Kock C, de Villiers KA, Smith PJ, Smith VJ, van Otterlo WA, Blackie MA. Jacobs L, et al. Among authors: de kock c, de villiers ka. ChemMedChem. 2015 Dec;10(12):2099-110. doi: 10.1002/cmdc.201500349. Epub 2015 Oct 8. ChemMedChem. 2015. PMID: 26447782

8

In vitro antiplasmodial activity of triazole-linked chloroquinoline derivatives synthesized from 7-chloro-N-(prop-2-yn-1-yl)quinolin-4-amine.

Taleli L, de Kock C, Smith PJ, Pelly SC, Blackie MAL, van Otterlo WAL. Taleli L, et al. Among authors: de kock c. Bioorg Med Chem. 2015 Aug 1;23(15):4163-4171. doi: 10.1016/j.bmc.2015.06.044. Epub 2015 Jun 27. Bioorg Med Chem. 2015. PMID: 26174655

9

Synthesis and evaluation of hybrid drugs for a potential HIV/AIDS-malaria combination therapy.

Aminake MN, Mahajan A, Kumar V, Hans R, Wiesner L, Taylor D, de Kock C, Grobler A, Smith PJ, Kirschner M, Rethwilm A, Pradel G, Chibale K. Aminake MN, et al. Among authors: de kock c. Bioorg Med Chem. 2012 Sep 1;20(17):5277-89. doi: 10.1016/j.bmc.2012.06.038. Epub 2012 Jun 29. Bioorg Med Chem. 2012. PMID: 22858300

10

UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria.

Brunschwig C, Lawrence N, Taylor D, Abay E, Njoroge M, Basarab GS, Le Manach C, Paquet T, Cabrera DG, Nchinda AT, de Kock C, Wiesner L, Denti P, Waterson D, Blasco B, Leroy D, Witty MJ, Donini C, Duffy J, Wittlin S, White KL, Charman SA, Jiménez-Díaz MB, Angulo-Barturen I, Herreros E, Gamo FJ, Rochford R, Mancama D, Coetzer TL, van der Watt ME, Reader J, Birkholtz LM, Marsh KC, Solapure SM, Burke JE, McPhail JA, Vanaerschot M, Fidock DA, Fish PV, Siegl P, Smith DA, Wirjanata G, Noviyanti R, Price RN, Marfurt J, Silue KD, Street LJ, Chibale K. Brunschwig C, et al. Among authors: de kock c. Antimicrob Agents Chemother. 2018 Aug 27;62(9):e00012-18. doi: 10.1128/AAC.00012-18. Print 2018 Sep. Antimicrob Agents Chemother. 2018. PMID: 29941635 Free PMC article.

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