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Cell-active carbazole derivatives as inhibitors of the zika virus protease.
Eur J Med Chem. 2019 Oct 15;180:536-545. doi: 10.1016/j.ejmech.2019.07.007. Epub 2019 Jul 17.
Eur J Med Chem. 2019.
PMID: 31344613
Amidoxime prodrugs convert to potent cell-active multimodal inhibitors of the dengue virus protease.
Swarbrick C, Zogali V, Chan KWK, Kiousis D, Gwee CP, Wang S, Lescar J, Luo D, von Itzstein M, Matsoukas MT, Panagiotakopoulos G, Vasudevan SG, Rassias G.
Swarbrick C, et al. Among authors: zogali v.
Eur J Med Chem. 2021 Nov 15;224:113695. doi: 10.1016/j.ejmech.2021.113695. Epub 2021 Jul 10.
Eur J Med Chem. 2021.
PMID: 34298282
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Carbazole to indolazepinone scaffold morphing leads to potent cell-active dengue antivirals.
Zogali V, Kiousis D, Voutyra S, Kalyva G, Abdul Mahid MB, Bist P, Ki Chan KW, Vasudevan SG, Rassias G.
Zogali V, et al.
Eur J Med Chem. 2024 Mar 15;268:116213. doi: 10.1016/j.ejmech.2024.116213. Epub 2024 Feb 16.
Eur J Med Chem. 2024.
PMID: 38382389
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