Yasushi Kohno - Search Results

Year	Number of Results
2007	1
2008	1
2009	1
2010	1
2011	6
2012	9
2013	3
2015	1
2016	3
2017	4
2020	2
2021	1
2024	0

1

Discovery of benzo[f]pyrido[4,3-b][1,4]oxazepin-10-one derivatives as orally available bromodomain and extra-terminal domain (BET) inhibitors with efficacy in an in vivo psoriatic animal model.

Sato M, Kondo T, Kohno Y, Seto S. Sato M, et al. Among authors: kohno y. Bioorg Med Chem. 2021 Mar 15;34:116015. doi: 10.1016/j.bmc.2021.116015. Epub 2021 Jan 25. Bioorg Med Chem. 2021. PMID: 33549905

2

Autofluorescence changes of tomato surface tissues during overripening.

Konagaya K, Riza DFA, Ogawa Y, Kohno Y, Kuramoto M, Takahashi N, Suzuki T, Kondo N. Konagaya K, et al. Among authors: kohno y. Photochem Photobiol Sci. 2020 Jul 1;19(7):879-884. doi: 10.1039/d0pp00125b. Epub 2020 Jun 24. Photochem Photobiol Sci. 2020. PMID: 32579662 Free article.

3

Discovery of BMS-986235/LAR-1219: A Potent Formyl Peptide Receptor 2 (FPR2) Selective Agonist for the Prevention of Heart Failure.

Asahina Y, Wurtz NR, Arakawa K, Carson N, Fujii K, Fukuchi K, Garcia R, Hsu MY, Ishiyama J, Ito B, Kick E, Lupisella J, Matsushima S, Ohata K, Ostrowski J, Saito Y, Tsuda K, Villarreal F, Yamada H, Yamaoka T, Wexler R, Gordon D, Kohno Y. Asahina Y, et al. Among authors: kohno y. J Med Chem. 2020 Sep 10;63(17):9003-9019. doi: 10.1021/acs.jmedchem.9b02101. Epub 2020 May 24. J Med Chem. 2020. PMID: 32407089

4

Discovery of novel pyrazolo[1,5-a]pyridine-based EP₁ receptor antagonists by scaffold hopping: Design, synthesis, and structure-activity relationships.

Nishigaya Y, Umei K, Saito Y, Watanabe H, Kondo T, Kondo A, Kawamura N, Tatani K, Kohno Y, Tanaka N, Seto S. Nishigaya Y, et al. Among authors: kohno y. Bioorg Med Chem Lett. 2017 Sep 1;27(17):4044-4050. doi: 10.1016/j.bmcl.2017.07.055. Epub 2017 Jul 25. Bioorg Med Chem Lett. 2017. PMID: 28784294

5

Identification of novel 1,2,3,6-tetrahydropyridyl-substituted benzo[d]thiazoles: Lead generation and optimization toward potent and orally active EP₁ receptor antagonists.

Umei K, Nishigaya Y, Tatani K, Kohno Y, Tanaka N, Seto S. Umei K, et al. Among authors: kohno y. Bioorg Med Chem. 2017 Jul 1;25(13):3406-3430. doi: 10.1016/j.bmc.2017.04.028. Epub 2017 Apr 26. Bioorg Med Chem. 2017. PMID: 28483455

6

Novel pyrazolo[1,5-a]pyridines as orally active EP₁ receptor antagonists: Synthesis, structure-activity relationship studies, and biological evaluation.

Umei K, Nishigaya Y, Kondo A, Tatani K, Tanaka N, Kohno Y, Seto S. Umei K, et al. Among authors: kohno y. Bioorg Med Chem. 2017 May 1;25(9):2635-2642. doi: 10.1016/j.bmc.2017.03.003. Epub 2017 Mar 14. Bioorg Med Chem. 2017. PMID: 28342692

7

Sulfonamide-based non-alkyne LpxC inhibitors as Gram-negative antibacterial agents.

Kawai T, Kazuhiko I, Takaya N, Yamaguchi Y, Kishii R, Kohno Y, Kurasaki H. Kawai T, et al. Among authors: kohno y. Bioorg Med Chem Lett. 2017 Feb 15;27(4):1045-1049. doi: 10.1016/j.bmcl.2016.12.059. Epub 2016 Dec 24. Bioorg Med Chem Lett. 2017. PMID: 28082037

8

LpxC Inhibitors: Design, Synthesis, and Biological Evaluation of Oxazolidinones as Gram-negative Antibacterial Agents.

Kurasaki H, Tsuda K, Shinoyama M, Takaya N, Yamaguchi Y, Kishii R, Iwase K, Ando N, Nomura M, Kohno Y. Kurasaki H, et al. Among authors: kohno y. ACS Med Chem Lett. 2016 Apr 5;7(6):623-8. doi: 10.1021/acsmedchemlett.6b00057. eCollection 2016 Jun 9. ACS Med Chem Lett. 2016. PMID: 27326338 Free PMC article.

9

Bitopic Sphingosine 1-Phosphate Receptor 3 (S1P3) Antagonist Rescue from Complete Heart Block: Pharmacological and Genetic Evidence for Direct S1P3 Regulation of Mouse Cardiac Conduction.

Sanna MG, Vincent KP, Repetto E, Nguyen N, Brown SJ, Abgaryan L, Riley SW, Leaf NB, Cahalan SM, Kiosses WB, Kohno Y, Brown JH, McCulloch AD, Rosen H, Gonzalez-Cabrera PJ. Sanna MG, et al. Among authors: kohno y. Mol Pharmacol. 2016 Jan;89(1):176-86. doi: 10.1124/mol.115.100222. Epub 2015 Oct 22. Mol Pharmacol. 2016. PMID: 26494861 Free PMC article.

10

Phosphodiesterase inhibitors. Part 6: design, synthesis, and structure-activity relationships of PDE4-inhibitory pyrazolo[1,5-a]pyridines with anti-inflammatory activity.

Kojima A, Takita S, Sumiya T, Ochiai K, Iwase K, Kishi T, Ohinata A, Yageta Y, Yasue T, Kohno Y. Kojima A, et al. Among authors: kohno y. Bioorg Med Chem Lett. 2013 Oct 1;23(19):5311-6. doi: 10.1016/j.bmcl.2013.07.069. Epub 2013 Aug 8. Bioorg Med Chem Lett. 2013. PMID: 23988356

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