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Page 1
Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate.
ACS Med Chem Lett. 2014 Feb 24;5(5):474-9. doi: 10.1021/ml400473x. eCollection 2014 May 8.
ACS Med Chem Lett. 2014.
PMID: 24900864
Free PMC article.
Evaluation and synthesis of polar aryl- and heteroaryl spiroazetidine-piperidine acetamides as ghrelin inverse agonists.
Orr ST, Beveridge R, Bhattacharya SK, Cameron KO, Coffey S, Fernando D, Hepworth D, Jackson MV, Khot V, Kosa R, Lapham K, Loria PM, McClure KF, Patel J, Rose C, Saenz J, Stock IA, Storer G, von Volkenburg M, Vrieze D, Wang G, Xiao J, Zhang Y.
Orr ST, et al. Among authors: vrieze d.
ACS Med Chem Lett. 2014 Dec 14;6(2):156-61. doi: 10.1021/ml500414n. eCollection 2015 Feb 12.
ACS Med Chem Lett. 2014.
PMID: 25699143
Free PMC article.
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Identification of (R)-6-(1-(4-cyano-3-methylphenyl)-5-cyclopentyl-4,5-dihydro-1H-pyrazol-3-yl)-2-methoxynicotinic acid, a highly potent and selective nonsteroidal mineralocorticoid receptor antagonist.
Casimiro-Garcia A, Piotrowski DW, Ambler C, Arhancet GB, Banker ME, Banks T, Boustany-Kari CM, Cai C, Chen X, Eudy R, Hepworth D, Hulford CA, Jennings SM, Loria PM, Meyers MJ, Petersen DN, Raheja NK, Sammons M, She L, Song K, Vrieze D, Wei L.
Casimiro-Garcia A, et al. Among authors: vrieze d.
J Med Chem. 2014 May 22;57(10):4273-88. doi: 10.1021/jm500206r. Epub 2014 Apr 30.
J Med Chem. 2014.
PMID: 24738581
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Synthesis and biological evaluation of amino-pyridines as androgen receptor antagonists for stimulating hair growth and reducing sebum production.
Hu LY, Lei HJ, Du D, Johnson TR, Fedij V, Kostlan C, Yue WS, Lovdahl M, Li JJ, Carroll M, Dettling D, Asbill J, Fan C, Wade K, Pocalyko D, Lapham K, Yalamanchili R, Samas B, Vrieze D, Ciotti S, Krieger-Burke T, Sliskovic D, Welgus H.
Hu LY, et al. Among authors: vrieze d.
Bioorg Med Chem Lett. 2007 Oct 15;17(20):5693-7. doi: 10.1016/j.bmcl.2007.07.059. Epub 2007 Aug 19.
Bioorg Med Chem Lett. 2007.
PMID: 17766112
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A highly enantioselective allylic amination reaction using a commercially available chiral rhodium catalyst: resolution of racemic allylic carbonates.
Vrieze DC, Hoge GS, Hoerter PZ, Van Haitsma JT, Samas BM.
Vrieze DC, et al.
Org Lett. 2009 Jul 16;11(14):3140-2. doi: 10.1021/ol901031b.
Org Lett. 2009.
PMID: 19527001
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Photochemical synthesis of 3-alkynals from 1-alkynoxy-9,10-anthraquinones.
Blankespoor RL, Boldenow PJ, Hansen EC, Kallemeyn JM, Lohse AG, Rubush DM, Vrieze D.
Blankespoor RL, et al. Among authors: vrieze d.
J Org Chem. 2009 May 15;74(10):3933-5. doi: 10.1021/jo900298y.
J Org Chem. 2009.
PMID: 19374382
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Diversity, Equity, and Inclusion Efforts at a Departmental Level: Building a Committee as a Vehicle for Advancing Progress.
Lingras KA, Alexander ME, Vrieze DM.
Lingras KA, et al. Among authors: vrieze dm.
J Clin Psychol Med Settings. 2023 Jun;30(2):356-379. doi: 10.1007/s10880-021-09809-w. Epub 2021 Sep 16.
J Clin Psychol Med Settings. 2023.
PMID: 34529234
Free PMC article.
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Tafamidis Treatment for Patients with Transthyretin Amyloid Cardiomyopathy.
Maurer MS, Schwartz JH, Gundapaneni B, Elliott PM, Merlini G, Waddington-Cruz M, Kristen AV, Grogan M, Witteles R, Damy T, Drachman BM, Shah SJ, Hanna M, Judge DP, Barsdorf AI, Huber P, Patterson TA, Riley S, Schumacher J, Stewart M, Sultan MB, Rapezzi C; ATTR-ACT Study Investigators.
Maurer MS, et al.
N Engl J Med. 2018 Sep 13;379(11):1007-1016. doi: 10.1056/NEJMoa1805689. Epub 2018 Aug 27.
N Engl J Med. 2018.
PMID: 30145929
Free article.
Clinical Trial.
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