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Pyridylpiperazine-based allosteric inhibitors of RND-type multidrug efflux pumps.
Nat Commun. 2022 Jan 10;13(1):115. doi: 10.1038/s41467-021-27726-2.
Nat Commun. 2022.
PMID: 35013254
Free PMC article.
On the Hunt for Next-Generation Antimicrobial Agents: An Online Symposium Organized Jointly by the French Society for Medicinal Chemistry (Société de Chimie Thérapeutique) and the French Microbiology Society (Société Française de Microbiologie) on 9-10 December 2021.
Antraygues K, Compagne N, Ruggieri F, Djaout K, Edoo Z, Eveque M, Faïon L, Gioia B, Tangara S, Vieira Da Cruz A, Villemagne B, Flipo M, Baulard A, Willand N.
Antraygues K, et al. Among authors: vieira da cruz a.
Pharmaceuticals (Basel). 2022 Mar 23;15(4):388. doi: 10.3390/ph15040388.
Pharmaceuticals (Basel). 2022.
PMID: 35455385
Free PMC article.
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Update on the Discovery of Efflux Pump Inhibitors against Critical Priority Gram-Negative Bacteria.
Compagne N, Vieira Da Cruz A, Müller RT, Hartkoorn RC, Flipo M, Pos KM.
Compagne N, et al. Among authors: vieira da cruz a.
Antibiotics (Basel). 2023 Jan 15;12(1):180. doi: 10.3390/antibiotics12010180.
Antibiotics (Basel). 2023.
PMID: 36671381
Free PMC article.
Review.
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Optimization of pyridylpiperazine-based inhibitors of the Escherichia coli AcrAB-TolC efflux pump.
Compagne N, Jiménez-Castellanos JC, Meurillon V, Pradel E, Vieira Da Cruz A, Piveteau C, Biela A, Eveque M, Leroux F, Deprez B, Willand N, Hartkoorn RC, Flipo M.
Compagne N, et al. Among authors: vieira da cruz a.
Eur J Med Chem. 2023 Nov 5;259:115630. doi: 10.1016/j.ejmech.2023.115630. Epub 2023 Jul 7.
Eur J Med Chem. 2023.
PMID: 37459793
Free article.
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Characterization of pyridylpiperazine-based efflux pump inhibitors for Acinetobacter baumannii.
Jiménez-Castellanos JC, Pradel E, Compagne N, Vieira Da Cruz A, Flipo M, Hartkoorn RC.
Jiménez-Castellanos JC, et al. Among authors: vieira da cruz a.
JAC Antimicrob Resist. 2023 Oct 24;5(5):dlad112. doi: 10.1093/jacamr/dlad112. eCollection 2023 Oct.
JAC Antimicrob Resist. 2023.
PMID: 37881353
Free PMC article.
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Polyhydroxylated Quinolizidine Iminosugars as Nanomolar Selective Inhibitors of α-Glucosidases.
Vieira Da Cruz A, Kanazawa A, Poisson JF, Behr JB, Py S.
Vieira Da Cruz A, et al.
J Org Chem. 2017 Sep 15;82(18):9866-9872. doi: 10.1021/acs.joc.7b01494. Epub 2017 Aug 28.
J Org Chem. 2017.
PMID: 28752763
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Pyridylpiperazine efflux pump inhibitor boosts in vivo antibiotic efficacy against K. pneumoniae.
Vieira Da Cruz A, Jiménez-Castellanos JC, Börnsen C, Van Maele L, Compagne N, Pradel E, Müller RT, Meurillon V, Soulard D, Piveteau C, Biela A, Dumont J, Leroux F, Deprez B, Willand N, Pos KM, Frangakis AS, Hartkoorn RC, Flipo M.
Vieira Da Cruz A, et al.
EMBO Mol Med. 2024 Jan;16(1):93-111. doi: 10.1038/s44321-023-00007-9. Epub 2023 Dec 20.
EMBO Mol Med. 2024.
PMID: 38177534
Free PMC article.
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