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Novel 3,4-isoxazolediamides as potent inhibitors of chaperone heat shock protein 90.
Baruchello R, Simoni D, Grisolia G, Barbato G, Marchetti P, Rondanin R, Mangiola S, Giannini G, Brunetti T, Alloatti D, Gallo G, Ciacci A, Vesci L, Castorina M, Milazzo FM, Cervoni ML, Guglielmi MB, Barbarino M, Foderà R, Pisano C, Cabri W. Baruchello R, et al. Among authors: vesci l. J Med Chem. 2011 Dec 22;54(24):8592-604. doi: 10.1021/jm201155e. Epub 2011 Nov 23. J Med Chem. 2011. PMID: 22066525
Natural and semisynthetic azaphilones as a new scaffold for Hsp90 inhibitors.
Musso L, Dallavalle S, Merlini L, Bava A, Nasini G, Penco S, Giannini G, Giommarelli C, De Cesare A, Zuco V, Vesci L, Pisano C, Castorina M, Milazzo F, Cervoni ML, Dal Piaz F, De Tommasi N, Zunino F. Musso L, et al. Among authors: vesci l. Bioorg Med Chem. 2010 Aug 15;18(16):6031-43. doi: 10.1016/j.bmc.2010.06.068. Epub 2010 Jul 1. Bioorg Med Chem. 2010. PMID: 20655237
New retinoid derivatives as back-ups of Adarotene.
Giannini G, Brunetti T, Battistuzzi G, Alloatti D, Quattrociocchi G, Cima MG, Merlini L, Dallavalle S, Cincinelli R, Nannei R, Vesci L, Bucci F, Foderà R, Guglielmi MB, Pisano C, Cabri W. Giannini G, et al. Among authors: vesci l. Bioorg Med Chem. 2012 Apr 1;20(7):2405-15. doi: 10.1016/j.bmc.2012.01.042. Epub 2012 Feb 6. Bioorg Med Chem. 2012. PMID: 22365912
Isoxazolo(aza)naphthoquinones: a new class of cytotoxic Hsp90 inhibitors.
Bargiotti A, Musso L, Dallavalle S, Merlini L, Gallo G, Ciacci A, Giannini G, Cabri W, Penco S, Vesci L, Castorina M, Milazzo FM, Cervoni ML, Barbarino M, Pisano C, Giommarelli C, Zuco V, De Cesare M, Zunino F. Bargiotti A, et al. Among authors: vesci l. Eur J Med Chem. 2012 Jul;53:64-75. doi: 10.1016/j.ejmech.2012.03.036. Epub 2012 Mar 28. Eur J Med Chem. 2012. PMID: 22538015
Camptothecins in tumor homing via an RGD sequence mimetic.
Alloatti D, Giannini G, Vesci L, Castorina M, Pisano C, Badaloni E, Cabri W. Alloatti D, et al. Among authors: vesci l. Bioorg Med Chem Lett. 2012 Oct 15;22(20):6509-12. doi: 10.1016/j.bmcl.2012.07.061. Epub 2012 Jul 26. Bioorg Med Chem Lett. 2012. PMID: 22959246
Novel PARP-1 inhibitors based on a 2-propanoyl-3H-quinazolin-4-one scaffold.
Giannini G, Battistuzzi G, Vesci L, Milazzo FM, De Paolis F, Barbarino M, Guglielmi MB, Carollo V, Gallo G, Artali R, Dallavalle S. Giannini G, et al. Among authors: vesci l. Bioorg Med Chem Lett. 2014 Jan 15;24(2):462-6. doi: 10.1016/j.bmcl.2013.12.048. Epub 2013 Dec 18. Bioorg Med Chem Lett. 2014. PMID: 24388690 Free article.
71 results