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Discovery and selection of TMC114, a next generation HIV-1 protease inhibitor.
J Med Chem. 2005 Mar 24;48(6):1813-22. doi: 10.1021/jm049560p.
J Med Chem. 2005.
PMID: 15771427
Design and optimization of tricyclic phtalimide analogues as novel inhibitors of HIV-1 integrase.
Verschueren WG, Dierynck I, Amssoms KI, Hu L, Boonants PM, Pille GM, Daeyaert FF, Hertogs K, Surleraux DL, Wigerinck PB.
Verschueren WG, et al.
J Med Chem. 2005 Mar 24;48(6):1930-40. doi: 10.1021/jm049559q.
J Med Chem. 2005.
PMID: 15771437
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Design of HIV-1 protease inhibitors active on multidrug-resistant virus.
Surleraux DL, de Kock HA, Verschueren WG, Pille GM, Maes LJ, Peeters A, Vendeville S, De Meyer S, Azijn H, Pauwels R, de Bethune MP, King NM, Prabu-Jeyabalan M, Schiffer CA, Wigerinck PB.
Surleraux DL, et al. Among authors: verschueren wg.
J Med Chem. 2005 Mar 24;48(6):1965-73. doi: 10.1021/jm049454n.
J Med Chem. 2005.
PMID: 15771440
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Synthesis and Evaluation of N-Phenyl-3-sulfamoyl-benzamide Derivatives as Capsid Assembly Modulators Inhibiting Hepatitis B Virus (HBV).
Vandyck K, Rombouts G, Stoops B, Tahri A, Vos A, Verschueren W, Wu Y, Yang J, Hou F, Huang B, Vergauwen K, Dehertogh P, Berke JM, Raboisson P.
Vandyck K, et al.
J Med Chem. 2018 Jul 26;61(14):6247-6260. doi: 10.1021/acs.jmedchem.8b00654. Epub 2018 Jul 3.
J Med Chem. 2018.
PMID: 29906396
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Design and synthesis of HIV-1 protease inhibitors for a long-acting injectable drug application.
Kesteleyn B, Amssoms K, Schepens W, Hache G, Verschueren W, Van De Vreken W, Rombauts K, Meurs G, Sterkens P, Stoops B, Baert L, Austin N, Wegner J, Masungi C, Dierynck I, Lundgren S, Jönsson D, Parkes K, Kalayanov G, Wallberg H, Rosenquist A, Samuelsson B, Van Emelen K, Thuring JW.
Kesteleyn B, et al.
Bioorg Med Chem Lett. 2013 Jan 1;23(1):310-7. doi: 10.1016/j.bmcl.2012.10.095. Epub 2012 Nov 1.
Bioorg Med Chem Lett. 2013.
PMID: 23177258
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