Design, synthesis and in vitro evaluation of novel SARS-CoV-2 3CLpro covalent inhibitors.
Stille JK, Tjutrins J, Wang G, Venegas FA, Hennecker C, Rueda AM, Sharon I, Blaine N, Miron CE, Pinus S, Labarre A, Plescia J, Burai Patrascu M, Zhang X, Wahba AS, Vlaho D, Huot MJ, Schmeing TM, Mittermaier AK, Moitessier N.
Stille JK, et al. Among authors: venegas fa.
Eur J Med Chem. 2022 Feb 5;229:114046. doi: 10.1016/j.ejmech.2021.114046. Epub 2021 Dec 11.
Eur J Med Chem. 2022.
PMID: 34995923
Free PMC article.