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Novel multi-target ligands of dopamine and serotonin receptors for the treatment of schizophrenia based on indazole and piperazine scaffolds-synthesis, biological activity, and structural evaluation.
Stępnicki P, Wronikowska-Denysiuk O, Zięba A, Targowska-Duda KM, Bartyzel A, Wróbel MZ, Wróbel TM, Szałaj K, Chodkowski A, Mirecka K, Budzyńska B, Fornal E, Turło J, Castro M, Kaczor AA. Stępnicki P, et al. Among authors: turlo j. J Enzyme Inhib Med Chem. 2023 Dec;38(1):2209828. doi: 10.1080/14756366.2023.2209828. J Enzyme Inhib Med Chem. 2023. PMID: 37184096 Free PMC article.
Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity: part 2.
Herold F, Izbicki Ł, Chodkowski A, Dawidowski M, Król M, Kleps J, Turło J, Wolska I, Nowak G, Stachowicz K, Dybała M, Siwek A, Nowak M, Pieniazek E, Jarończyk M, Sylte I, Mazurek AP. Herold F, et al. Among authors: turlo j. Eur J Med Chem. 2009 Nov;44(11):4702-15. doi: 10.1016/j.ejmech.2009.07.007. Epub 2009 Jul 16. Eur J Med Chem. 2009. PMID: 19665823
Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT(1A) activity. part 3.
Herold F, Chodkowski A, Izbicki Ł, Turło J, Dawidowski M, Kleps J, Nowak G, Stachowicz K, Dybała M, Siwek A, Mazurek AP, Mazurek A, Pluciński F. Herold F, et al. Among authors: turlo j. Eur J Med Chem. 2011 Jan;46(1):142-9. doi: 10.1016/j.ejmech.2010.10.026. Epub 2010 Oct 29. Eur J Med Chem. 2011. PMID: 21093118
Synthesis and biological evaluation of novel pyrrolidine-2,5-dione derivatives as potential antidepressant agents. Part 1.
Wróbel MZ, Chodkowski A, Herold F, Gomółka A, Kleps J, Mazurek AP, Pluciński F, Mazurek A, Nowak G, Siwek A, Stachowicz K, Sławińska A, Wolak M, Szewczyk B, Satała G, Bojarski AJ, Turło J. Wróbel MZ, et al. Among authors: turlo j. Eur J Med Chem. 2013 May;63:484-500. doi: 10.1016/j.ejmech.2013.02.033. Epub 2013 Mar 5. Eur J Med Chem. 2013. PMID: 23524160
Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT(1A) activity. Part 5.
Gomółka A, Ciesielska A, Wróbel MZ, Chodkowski A, Kleps J, Dawidowski M, Siwek A, Wolak M, Stachowicz K, Sławińska A, Nowak G, Satała G, Bojarski AJ, Belka M, Ulenberg S, Bączek T, Skowronek P, Turło J, Herold F. Gomółka A, et al. Among authors: turlo j. Eur J Med Chem. 2015 Jun 15;98:221-36. doi: 10.1016/j.ejmech.2015.05.003. Epub 2015 May 9. Eur J Med Chem. 2015. PMID: 26043160
61 results