Tardugno M - Search Results

1

Gold drug auranofin restricts the viral reservoir in the monkey AIDS model and induces containment of viral load following ART suspension.

Lewis MG, DaFonseca S, Chomont N, Palamara AT, Tardugno M, Mai A, Collins M, Wagner WL, Yalley-Ogunro J, Greenhouse J, Chirullo B, Norelli S, Garaci E, Savarino A. Lewis MG, et al. Among authors: tardugno m. AIDS. 2011 Jul 17;25(11):1347-56. doi: 10.1097/QAD.0b013e328347bd77. AIDS. 2011. PMID: 21505294

2

Pyrrole-based hydroxamates and 2-aminoanilides: histone deacetylase inhibition and cellular activities.

Valente S, Conte M, Tardugno M, Massa S, Nebbioso A, Altucci L, Mai A. Valente S, et al. Among authors: tardugno m. ChemMedChem. 2009 Sep;4(9):1411-5. doi: 10.1002/cmdc.200900082. ChemMedChem. 2009. PMID: 19504533 No abstract available.

3

Novel uracil-based 2-aminoanilide and 2-aminoanilide-like derivatives: histone deacetylase inhibition and in-cell activities.

Mai A, Perrone A, Nebbioso A, Rotili D, Valente S, Tardugno M, Massa S, De Bellis F, Altucci L. Mai A, et al. Among authors: tardugno m. Bioorg Med Chem Lett. 2008 Apr 15;18(8):2530-5. doi: 10.1016/j.bmcl.2008.03.055. Epub 2008 Mar 22. Bioorg Med Chem Lett. 2008. PMID: 18381238

4

Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.

Valente S, Lepore I, Dell'Aversana C, Tardugno M, Castellano S, Sbardella G, Tomassi S, Di Maro S, Novellino E, Di Santo R, Costi R, Altucci L, Mai A. Valente S, et al. Among authors: tardugno m. Biochimie. 2012 Nov;94(11):2308-13. doi: 10.1016/j.biochi.2012.06.003. Epub 2012 Jun 16. Biochimie. 2012. PMID: 22709867

5

Study of 1,4-dihydropyridine structural scaffold: discovery of novel sirtuin activators and inhibitors.

Mai A, Valente S, Meade S, Carafa V, Tardugno M, Nebbioso A, Galmozzi A, Mitro N, De Fabiani E, Altucci L, Kazantsev A. Mai A, et al. Among authors: tardugno m. J Med Chem. 2009 Sep 10;52(17):5496-504. doi: 10.1021/jm9008289. J Med Chem. 2009. PMID: 19663498

6

Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells.

Valente S, Liu Y, Schnekenburger M, Zwergel C, Cosconati S, Gros C, Tardugno M, Labella D, Florean C, Minden S, Hashimoto H, Chang Y, Zhang X, Kirsch G, Novellino E, Arimondo PB, Miele E, Ferretti E, Gulino A, Diederich M, Cheng X, Mai A. Valente S, et al. Among authors: tardugno m. J Med Chem. 2014 Feb 13;57(3):701-13. doi: 10.1021/jm4012627. Epub 2014 Jan 15. J Med Chem. 2014. PMID: 24387159 Free PMC article.

7

Novel cinnamyl hydroxyamides and 2-aminoanilides as histone deacetylase inhibitors: apoptotic induction and cytodifferentiation activity.

Valente S, Tardugno M, Conte M, Cirilli R, Perrone A, Ragno R, Simeoni S, Tramontano A, Massa S, Nebbioso A, Miceli M, Franci G, Brosch G, Altucci L, Mai A. Valente S, et al. Among authors: tardugno m. ChemMedChem. 2011 Apr 4;6(4):698-712. doi: 10.1002/cmdc.201000535. Epub 2011 Mar 4. ChemMedChem. 2011. PMID: 21374822

8

1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells.

Valente S, Mellini P, Spallotta F, Carafa V, Nebbioso A, Polletta L, Carnevale I, Saladini S, Trisciuoglio D, Gabellini C, Tardugno M, Zwergel C, Cencioni C, Atlante S, Moniot S, Steegborn C, Budriesi R, Tafani M, Del Bufalo D, Altucci L, Gaetano C, Mai A. Valente S, et al. Among authors: tardugno m. J Med Chem. 2016 Feb 25;59(4):1471-91. doi: 10.1021/acs.jmedchem.5b01117. Epub 2016 Jan 5. J Med Chem. 2016. PMID: 26689352

9

Biochemical, structural, and biological evaluation of tranylcypromine derivatives as inhibitors of histone demethylases LSD1 and LSD2.

Binda C, Valente S, Romanenghi M, Pilotto S, Cirilli R, Karytinos A, Ciossani G, Botrugno OA, Forneris F, Tardugno M, Edmondson DE, Minucci S, Mattevi A, Mai A. Binda C, et al. Among authors: tardugno m. J Am Chem Soc. 2010 May 19;132(19):6827-33. doi: 10.1021/ja101557k. J Am Chem Soc. 2010. PMID: 20415477

10

Protein recognition by short peptide reversible inhibitors of the chromatin-modifying LSD1/CoREST lysine demethylase.

Tortorici M, Borrello MT, Tardugno M, Chiarelli LR, Pilotto S, Ciossani G, Vellore NA, Bailey SG, Cowan J, O'Connell M, Crabb SJ, Packham G, Mai A, Baron R, Ganesan A, Mattevi A. Tortorici M, et al. Among authors: tardugno m. ACS Chem Biol. 2013 Aug 16;8(8):1677-82. doi: 10.1021/cb4001926. Epub 2013 Jun 11. ACS Chem Biol. 2013. PMID: 23721412

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

17 results

Search Page