Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring.
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Kanada R, et al. Among authors: takahashi m.
Bioorg Med Chem Lett. 2022 Jun 15;66:128726. doi: 10.1016/j.bmcl.2022.128726. Epub 2022 Apr 9.
Bioorg Med Chem Lett. 2022.
PMID: 35413416