Spetea M - Search Results

1

Opioids and Their Receptors: Present and Emerging Concepts in Opioid Drug Discovery II.

Van Rijn RM, Spetea M. Van Rijn RM, et al. Among authors: spetea m. Molecules. 2022 May 13;27(10):3140. doi: 10.3390/molecules27103140. Molecules. 2022. PMID: 35630616 Free PMC article.

2

Synthesis and pharmacological activities of 6-glycine substituted 14-phenylpropoxymorphinans, a novel class of opioids with high opioid receptor affinities and antinociceptive potencies.

Spetea M, Windisch P, Guo Y, Bileviciute-Ljungar I, Schütz J, Asim MF, Berzetei-Gurske IP, Riba P, Kiraly K, Fürst S, Al-Khrasani M, Schmidhammer H. Spetea M, et al. J Med Chem. 2011 Feb 24;54(4):980-8. doi: 10.1021/jm101211p. Epub 2011 Jan 14. J Med Chem. 2011. PMID: 21235243 Free PMC article.

3

Recent advances in the development of 14-alkoxy substituted morphinans as potent and safer opioid analgesics.

Spetea M, Schmidhammer H. Spetea M, et al. Curr Med Chem. 2012;19(15):2442-57. doi: 10.2174/092986712800269308. Curr Med Chem. 2012. PMID: 22455592 Review.

4

Discovery and pharmacological evaluation of a diphenethylamine derivative (HS665), a highly potent and selective κ opioid receptor agonist.

Spetea M, Berzetei-Gurske IP, Guerrieri E, Schmidhammer H. Spetea M, et al. J Med Chem. 2012 Nov 26;55(22):10302-6. doi: 10.1021/jm301258w. Epub 2012 Nov 7. J Med Chem. 2012. PMID: 23134120

5

Current κ opioid receptor ligands and discovery of a new molecular scaffold as a κ opioid receptor antagonist using pharmacophore-based virtual screening.

Spetea M, Asim MF, Noha S, Wolber G, Schmidhammer H. Spetea M, et al. Curr Pharm Des. 2013;19(42):7362-72. doi: 10.2174/138161281942140105162601. Curr Pharm Des. 2013. PMID: 23448472

6

The µ opioid receptor and ligands acting at the µ opioid receptor, as therapeutics and potential therapeutics.

Spetea M, Asim MF, Wolber G, Schmidhammer H. Spetea M, et al. Curr Pharm Des. 2013;19(42):7415-34. doi: 10.2174/13816128113199990362. Curr Pharm Des. 2013. PMID: 23448479 Review.

7

Opioid receptors and their ligands in the musculoskeletal system and relevance for pain control.

Spetea M. Spetea M. Curr Pharm Des. 2013;19(42):7382-90. doi: 10.2174/13816128113199990363. Curr Pharm Des. 2013. PMID: 23448480 Review.

8

Synthesis and pharmacological evaluation of [(3)H]HS665, a novel, highly selective radioligand for the kappa opioid receptor.

Guerrieri E, Mallareddy JR, Tóth G, Schmidhammer H, Spetea M. Guerrieri E, et al. Among authors: spetea m. ACS Chem Neurosci. 2015 Mar 18;6(3):456-63. doi: 10.1021/cn5002792. Epub 2014 Dec 24. ACS Chem Neurosci. 2015. PMID: 25496417

9

Highly Potent and Selective New Diphenethylamines Interacting with the κ-Opioid Receptor: Synthesis, Pharmacology, and Structure-Activity Relationships.

Erli F, Guerrieri E, Ben Haddou T, Lantero A, Mairegger M, Schmidhammer H, Spetea M. Erli F, et al. Among authors: spetea m. J Med Chem. 2017 Sep 14;60(17):7579-7590. doi: 10.1021/acs.jmedchem.7b00981. Epub 2017 Aug 30. J Med Chem. 2017. PMID: 28825813 Free PMC article.

10

A bifunctional-biased mu-opioid agonist-neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects.

Drieu la Rochelle A, Guillemyn K, Dumitrascuta M, Martin C, Utard V, Quillet R, Schneider S, Daubeuf F, Willemse T, Mampuys P, Maes BUW, Frossard N, Bihel F, Spetea M, Simonin F, Ballet S. Drieu la Rochelle A, et al. Among authors: spetea m. Pain. 2018 Sep;159(9):1705-1718. doi: 10.1097/j.pain.0000000000001262. Pain. 2018. PMID: 29708942

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