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Enterovirus inhibitory activity of C-8-tert-butyl substituted 4-aryl-6,7,8,9-tetrahydrobenzo[4,5]thieno[3,2-e][1,2,4]triazolo[4,3-a]pyrimidin-5(4H)-ones.
Bioorg Med Chem Lett. 2017 Aug 1;27(15):3582-3585. doi: 10.1016/j.bmcl.2017.05.030. Epub 2017 May 19.
Bioorg Med Chem Lett. 2017.
PMID: 28587824
Enteroviral replication inhibition by N-Alkyl triazolopyrimidinone derivatives through a non-capsid binding mode.
Kumar Biswas B, Soo Shin J, Malpani YR, Hwang D, Jung E, Bong Han S, Vishakantegowda AG, Jung YS.
Kumar Biswas B, et al. Among authors: soo shin j.
Bioorg Med Chem Lett. 2022 May 15;64:128673. doi: 10.1016/j.bmcl.2022.128673. Epub 2022 Mar 12.
Bioorg Med Chem Lett. 2022.
PMID: 35292344
Free article.
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Discovery of (E)-2-(hydroxyimino)-N-(2 ((4methylpentyl)amino)ethyl)acetamide (KR-27425) as a non-pyridinium oxime reactivator of paraoxon-inhibited acetylcholinesterase.
Vishakantegowda AG, Girmay BS, Shin JS, Lee JY, Ahn S, Jung YS.
Vishakantegowda AG, et al.
Bioorg Med Chem Lett. 2023 Nov 15;96:129504. doi: 10.1016/j.bmcl.2023.129504. Epub 2023 Oct 12.
Bioorg Med Chem Lett. 2023.
PMID: 37838342
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Strong transcription blockage mediated by R-loop formation within a G-rich homopurine-homopyrimidine sequence localized in the vicinity of the promoter.
Belotserkovskii BP, Soo Shin JH, Hanawalt PC.
Belotserkovskii BP, et al. Among authors: soo shin jh.
Nucleic Acids Res. 2017 Jun 20;45(11):6589-6599. doi: 10.1093/nar/gkx403.
Nucleic Acids Res. 2017.
PMID: 28498974
Free PMC article.
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