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Methods of Synthesis and Antiviral Activity of New 4-Alkyl-3-Nitro-1,4-Dihydroazolo[5,1-c][1,2,4]Triazin-4-ols.
Drokin RA, Tiufiakov DV, Voinkov EK, Slepukhin PA, Ulomsky EN, Esaulkova YL, Volobueva AS, Lantseva KS, Misyurina MA, Zarubaev VV, Rusinov VL. Drokin RA, et al. Among authors: slepukhin pa. Chem Heterocycl Compd (N Y). 2021;57(4):473-478. doi: 10.1007/s10593-021-02926-2. Epub 2021 May 12. Chem Heterocycl Compd (N Y). 2021. PMID: 33994554 Free PMC article.
6-Nitroazolo[1,5-a]pyrimidin-7(4H)-ones as Antidiabetic Agents.
Spasov AA, Babkov DA, Sysoeva VA, Litvinov RA, Shamshina DD, Ulomsky EN, Savateev KV, Fedotov VV, Slepukhin PA, Chupakhin ON, Charushin VN, Rusinov VL. Spasov AA, et al. Among authors: slepukhin pa. Arch Pharm (Weinheim). 2017 Dec;350(12). doi: 10.1002/ardp.201700226. Epub 2017 Nov 20. Arch Pharm (Weinheim). 2017. PMID: 29152780
15N-Labelling and structure determination of adamantylated azolo-azines in solution.
Deev SL, Paramonov AS, Shestakova TS, Khalymbadzha IA, Chupakhin ON, Subbotina JO, Eltsov OS, Slepukhin PA, Rusinov VL, Arseniev AS, Shenkarev ZO. Deev SL, et al. Among authors: slepukhin pa. Beilstein J Org Chem. 2017 Nov 29;13:2535-2548. doi: 10.3762/bjoc.13.250. eCollection 2017. Beilstein J Org Chem. 2017. PMID: 29259663 Free PMC article.
Nitrothiadiazolo[3,2-a]pyrimidines as promising antiglycating agents.
Savateev K, Fedotov V, Butorin I, Eltsov O, Slepukhin P, Ulomsky E, Rusinov V, Litvinov R, Babkov D, Khokhlacheva E, Radaev P, Vassiliev P, Spasov A. Savateev K, et al. Eur J Med Chem. 2020 Jan 1;185:111808. doi: 10.1016/j.ejmech.2019.111808. Epub 2019 Oct 25. Eur J Med Chem. 2020. PMID: 31683103
Synthesis and antiviral activity of nonannulated tetrazolylpyrimidines.
Ostrovskii VА, Danagulyan GG, Nesterova OM, Pavlyukova YN, Tolstyakov VV, Zarubina OS, Slepukhin PА, Esaulkova YL, Muryleva AА, Zarubaev VV, Trifonov RE. Ostrovskii VА, et al. Chem Heterocycl Compd (N Y). 2021;57(4):448-454. doi: 10.1007/s10593-021-02922-6. Epub 2021 May 14. Chem Heterocycl Compd (N Y). 2021. PMID: 34007083 Free PMC article.
New heteroanalogs of tricyclic ascidian alkaloids: synthesis and biological activity.
Goryaeva MV, Kushch SO, Burgart YV, Ezhikova MA, Kodess MI, Slepukhin PA, Triandafilova GA, Krasnykh OP, Yakovleva EI, Zarubaev VV, Sinegubova EO, Esaulkova IL, Shtro AA, Galochkina AV, Nikolaeva YV, Saloutin VI. Goryaeva MV, et al. Among authors: slepukhin pa. Org Biomol Chem. 2021 Nov 25;19(45):9925-9935. doi: 10.1039/d1ob01843d. Org Biomol Chem. 2021. PMID: 34735561
4-(Aryl)-Benzo[4,5]imidazo[1,2-a]pyrimidine-3-Carbonitrile-Based Fluorophores: Povarov Reaction-Based Synthesis, Photophysical Studies, and DFT Calculations.
Fedotov VV, Valieva MI, Taniya OS, Aminov SV, Kharitonov MA, Novikov AS, Kopchuk DS, Slepukhin PA, Zyryanov GV, Ulomsky EN, Rusinov VL, Charushin VN. Fedotov VV, et al. Among authors: slepukhin pa. Molecules. 2022 Nov 19;27(22):8029. doi: 10.3390/molecules27228029. Molecules. 2022. PMID: 36432130 Free PMC article.
Functionalization, cyclization and antiviral activity of A-secotriterpenoids.
Grishko VV, Galaiko NV, Tolmacheva IA, Kucherov II, Eremin VF, Boreko EI, Savinova OV, Slepukhin PA. Grishko VV, et al. Among authors: slepukhin pa. Eur J Med Chem. 2014 Aug 18;83:601-8. doi: 10.1016/j.ejmech.2013.12.058. Epub 2014 Jan 10. Eur J Med Chem. 2014. PMID: 24997292
47 results