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Inhibition of the norA gene expression and the NorA efflux pump by the tannic acid.
Tintino SR, Wilairatana P, de Souza VCA, da Silva JMA, Pereira PS, de Morais Oliveira-Tintino CD, de Matos YMLS, Júnior JTC, de Queiroz Balbino V, Siqueira-Junior JP, Menezes IRA, Siyadatpanah A, Coutinho HDM, Balbino TCL. Tintino SR, et al. Among authors: siqueira junior jp. Sci Rep. 2023 Oct 13;13(1):17394. doi: 10.1038/s41598-023-43038-5. Sci Rep. 2023. PMID: 37833301 Free PMC article.
Preclinical development of kinetin as a safe error-prone SARS-CoV-2 antiviral able to attenuate virus-induced inflammation.
Souza TML, Pinho VD, Setim CF, Sacramento CQ, Marcon R, Fintelman-Rodrigues N, Chaves OA, Heller M, Temerozo JR, Ferreira AC, Mattos M, Momo PB, Dias SSG, Gesto JSM, Pereira-Dutra F, Viola JPB, Queiroz-Junior CM, Guimarães LC, Chaves IM, Guimarães PPG, Costa VV, Teixeira MM, Bou-Habib DC, Bozza PT, Aguillón AR, Siqueira-Junior J, Macedo-Junior S, Andrade EL, Fadanni GP, Tolouei SEL, Potrich FB, Santos AA, Marques NF, Calixto JB, Rabi JA. Souza TML, et al. Among authors: siqueira junior j. Nat Commun. 2023 Jan 13;14(1):199. doi: 10.1038/s41467-023-35928-z. Nat Commun. 2023. PMID: 36639383 Free PMC article.
Enhancement of the antibiotic activity by quercetin against Staphylococcus aureus efflux pumps.
Dos Santos JFS, Tintino SR, da Silva ARP, Dos S Barbosa CR, Scherf JR, de S Silveira Z, de Freitas TS, de Lacerda Neto LJ, Barros LM, de A Menezes IR, Coutinho HDM, Siqueira-Júnior JP, Cunha FAB. Dos Santos JFS, et al. Among authors: siqueira junior jp. J Bioenerg Biomembr. 2021 Apr;53(2):157-167. doi: 10.1007/s10863-021-09886-4. Epub 2021 Mar 8. J Bioenerg Biomembr. 2021. PMID: 33683535
Aminophenyl chalcones potentiating antibiotic activity and inhibiting bacterial efflux pump.
Siqueira MMR, Freire PTC, Cruz BG, de Freitas TS, Bandeira PN, Silva Dos Santos H, Nogueira CES, Teixeira AMR, Pereira RLS, Xavier JDC, Campina FF, Dos Santos Barbosa CR, Neto JBA, da Silva MMC, Siqueira-Júnior JP, Douglas Melo Coutinho H. Siqueira MMR, et al. Among authors: siqueira junior jp. Eur J Pharm Sci. 2021 Mar 1;158:105695. doi: 10.1016/j.ejps.2020.105695. Epub 2020 Dec 29. Eur J Pharm Sci. 2021. PMID: 33383131
Inhibition of the NorA efflux pump of S. aureus by (Z)-5-(4-Fluorobenzylidene)-Imidazolidines.
Faillace MS, Alves Borges Leal AL, Araújo de Oliveira Alcântara F, Ferreira JHL, de Siqueira-Júnior JP, Sampaio Nogueira CE, Barreto HM, Peláez WJ. Faillace MS, et al. Among authors: de siqueira junior jp. Bioorg Med Chem Lett. 2021 Jan 1;31:127670. doi: 10.1016/j.bmcl.2020.127670. Epub 2020 Nov 6. Bioorg Med Chem Lett. 2021. PMID: 33161124
Prevention and control of Aedes transmitted infections in the post-pandemic scenario of COVID-19: challenges and opportunities for the region of the Americas.
Dantés HG, Manrique-Saide P, Vazquez-Prokopec G, Morales FC, Siqueira Junior JB, Pimenta F, Coelho G, Bezerra H. Dantés HG, et al. Among authors: siqueira junior jb. Mem Inst Oswaldo Cruz. 2020;115:e200284. doi: 10.1590/0074-02760200284. Epub 2020 Aug 5. Mem Inst Oswaldo Cruz. 2020. PMID: 32785481 Free PMC article.
85 results