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Page 1
Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease.
Makhaeva GF, Kovaleva NV, Rudakova EV, Boltneva NP, Grishchenko MV, Lushchekina SV, Astakhova TY, Serebryakova OG, Timokhina EN, Zhilina EF, Shchegolkov EV, Ulitko MV, Radchenko EV, Palyulin VA, Burgart YV, Saloutin VI, Bachurin SO, Richardson RJ. Makhaeva GF, et al. Among authors: shchegolkov ev. Int J Mol Sci. 2023 Jan 24;24(3):2285. doi: 10.3390/ijms24032285. Int J Mol Sci. 2023. PMID: 36768608 Free PMC article.
Synthesis, molecular docking, and biological activity of polyfluoroalkyl dihydroazolo[5,1-c][1,2,4]triazines as selective carboxylesterase inhibitors.
Shchegol'kov EV, Makhaeva GF, Boltneva NP, Lushchekina SV, Serebryakova OG, Rudakova EV, Kovaleva NV, Burgart YV, Saloutin VI, Chupakhin ON, Bachurin SO, Richardson RJ. Shchegol'kov EV, et al. Bioorg Med Chem. 2017 Aug 1;25(15):3997-4007. doi: 10.1016/j.bmc.2017.05.045. Epub 2017 May 20. Bioorg Med Chem. 2017. PMID: 28578994
Synthesis, molecular docking, and biological evaluation of 3-oxo-2-tolylhydrazinylidene-4,4,4-trifluorobutanoates bearing higher and natural alcohol moieties as new selective carboxylesterase inhibitors.
Makhaeva GF, Elkina NA, Shchegolkov EV, Boltneva NP, Lushchekina SV, Serebryakova OG, Rudakova EV, Kovaleva NV, Radchenko EV, Palyulin VA, Burgart YV, Saloutin VI, Bachurin SO, Richardson RJ. Makhaeva GF, et al. Among authors: shchegolkov ev. Bioorg Chem. 2019 Oct;91:103097. doi: 10.1016/j.bioorg.2019.103097. Epub 2019 Jul 3. Bioorg Chem. 2019. PMID: 31323527
Synthesis of 2-arylhydrazinylidene-3-oxo-4,4,4-trifluorobutanoic acids as new selective carboxylesterase inhibitors and radical scavengers.
Khudina OG, Makhaeva GF, Elkina NA, Boltneva NP, Serebryakova OG, Shchegolkov EV, Rudakova EV, Lushchekina SV, Burgart YV, Bachurin SO, Richardson RJ, Saloutin VI. Khudina OG, et al. Among authors: shchegolkov ev. Bioorg Med Chem Lett. 2019 Dec 1;29(23):126716. doi: 10.1016/j.bmcl.2019.126716. Epub 2019 Oct 14. Bioorg Med Chem Lett. 2019. PMID: 31640885
Multiple biological active 4-aminopyrazoles containing trifluoromethyl and their 4-nitroso-precursors: Synthesis and evaluation.
Burgart YV, Agafonova NA, Shchegolkov EV, Krasnykh OP, Kushch SO, Evstigneeva NP, Gerasimova NA, Maslova VV, Triandafilova GA, Solodnikov SY, Ulitko MV, Makhaeva GF, Rudakova EV, Borisevich SS, Zilberberg NV, Kungurov NV, Saloutin VI, Chupakhin ON. Burgart YV, et al. Among authors: shchegolkov ev. Eur J Med Chem. 2020 Dec 15;208:112768. doi: 10.1016/j.ejmech.2020.112768. Epub 2020 Aug 23. Eur J Med Chem. 2020. PMID: 32932211
Novel potent bifunctional carboxylesterase inhibitors based on a polyfluoroalkyl-2-imino-1,3-dione scaffold.
Makhaeva GF, Lushchekina SV, Boltneva NP, Serebryakova OG, Kovaleva NV, Rudakova EV, Elkina NA, Shchegolkov EV, Burgart YV, Stupina TS, Terentiev AA, Radchenko EV, Palyulin VA, Saloutin VI, Bachurin SO, Richardson RJ. Makhaeva GF, et al. Among authors: shchegolkov ev. Eur J Med Chem. 2021 Jun 5;218:113385. doi: 10.1016/j.ejmech.2021.113385. Epub 2021 Mar 15. Eur J Med Chem. 2021. PMID: 33831780
18 results