Skip to main page content
U.S. flag

An official website of the United States government

Dot gov

The .gov means it’s official.
Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you’re on a federal government site.

Https

The site is secure.
The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.

Access keys NCBI Homepage MyNCBI Homepage Main Content Main Navigation

Search Page

Filters

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

Search Results

12 results

Filters applied: . Clear all
Results are displayed in a computed author sort order. The Results By Year timeline is not available.
Page 1
Novel Copper-Containing Cytotoxic Agents Based on 2-Thioxoimidazolones.
Krasnovskaya OO, Guk DA, Naumov AE, Nikitina VN, Semkina AS, Vlasova KY, Pokrovsky V, Ryabaya OO, Karshieva SS, Skvortsov DA, Zhirkina IV, Shafikov RR, Gorelkin PV, Vaneev AN, Erofeev AS, Mazur DM, Tafeenko VA, Pergushov VI, Melnikov MY, Soldatov MA, Shapovalov VV, Soldatov AV, Akasov RA, Gerasimov VM, Sakharov DA, Moiseeva AA, Zyk NV, Beloglazkina EK, Majouga AG. Krasnovskaya OO, et al. Among authors: shafikov rr. J Med Chem. 2020 Nov 12;63(21):13031-13063. doi: 10.1021/acs.jmedchem.0c01196. Epub 2020 Oct 20. J Med Chem. 2020. PMID: 32985193
New ferrocene-based 2-thio-imidazol-4-ones and their copper complexes. Synthesis and cytotoxicity.
Guk DA, Krasnovskaya OO, Dashkova NS, Skvortsov DA, Rubtsova MP, Dyadchenko VP, Yudina ES, Kosarev MA, Soldatov AV, Shapovalov VV, Semkina AS, Vlasova KY, Pergushov VI, Shafikov RR, Moiseeva AA, Andreeva AV, Andreeva AA, Melnikov MY, Zyk NV, Majouga AG, Beloglazkina EK. Guk DA, et al. Among authors: shafikov rr. Dalton Trans. 2018 Dec 11;47(48):17357-17366. doi: 10.1039/c8dt03164a. Dalton Trans. 2018. PMID: 30480670
Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them.
Machulkin AE, Shafikov RR, Uspenskaya AA, Petrov SA, Ber AP, Skvortsov DA, Nimenko EA, Zyk NU, Smirnova GB, Pokrovsky VS, Abakumov MA, Saltykova IV, Akhmirov RT, Garanina AS, Polshakov VI, Saveliev OY, Ivanenkov YA, Aladinskaya AV, Finko AV, Yamansarov EU, Krasnovskaya OO, Erofeev AS, Gorelkin PV, Dontsova OA, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: shafikov rr. J Med Chem. 2021 Apr 22;64(8):4532-4552. doi: 10.1021/acs.jmedchem.0c01935. Epub 2021 Apr 6. J Med Chem. 2021. PMID: 33822606
PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation.
Machulkin AE, Uspenskaya AA, Zyk NY, Nimenko EA, Ber AP, Petrov SA, Shafikov RR, Skvortsov DA, Smirnova GB, Borisova YA, Pokrovsky VS, Kolmogorov VS, Vaneev AN, Ivanenkov YA, Khudyakov AD, Kovalev SV, Erofeev AS, Gorelkin PV, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: shafikov rr. Eur J Med Chem. 2022 Jan 5;227:113936. doi: 10.1016/j.ejmech.2021.113936. Epub 2021 Oct 23. Eur J Med Chem. 2022. PMID: 34717125
Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate.
Machulkin AE, Uspenskaya AA, Zyk NU, Nimenko EA, Ber AP, Petrov SA, Polshakov VI, Shafikov RR, Skvortsov DA, Plotnikova EA, Pankratov AA, Smirnova GB, Borisova YA, Pokrovsky VS, Kolmogorov VS, Vaneev AN, Khudyakov AD, Chepikova OE, Kovalev S, Zamyatnin AA Jr, Erofeev A, Gorelkin P, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: shafikov rr. J Med Chem. 2021 Dec 9;64(23):17123-17145. doi: 10.1021/acs.jmedchem.1c01157. Epub 2021 Nov 19. J Med Chem. 2021. PMID: 34797052
Correction: New ferrocene-based 2-thio-imidazol-4-ones and their copper complexes. Synthesis and cytotoxicity.
Guk DA, Krasnovskaya OO, Dashkova NS, Skvortsov DA, Rubtsova MP, Dyadchenko VP, Yudina ES, Kosarev MA, Soldatov AV, Shapovalov VV, Semkina AS, Vlasova KY, Pergushov VI, Shafikov RR, Moiseeva AA, Andreeva AV, Melnikov MY, Zyk NV, Majouga AG, Beloglazkina EK. Guk DA, et al. Among authors: shafikov rr. Dalton Trans. 2019 Jan 2;48(2):752. doi: 10.1039/c8dt90222d. Dalton Trans. 2019. PMID: 30542689
New copper(II) thiohydantoin complexes: Synthesis, characterization, and assessment of their interaction with bovine serum albumin and DNA.
Tishchenko K, Beloglazkina E, Proskurnin M, Malinnikov V, Guk D, Muratova M, Krasnovskaya O, Udina A, Skvortsov D, Shafikov RR, Ivanenkov Y, Aladinskiy V, Sorokin I, Gromov O, Majouga A, Zyk N. Tishchenko K, et al. Among authors: shafikov rr. J Inorg Biochem. 2017 Oct;175:190-197. doi: 10.1016/j.jinorgbio.2017.07.015. Epub 2017 Jul 21. J Inorg Biochem. 2017. PMID: 28756175
Synthesis and biological evaluation of PSMA-targeting paclitaxel conjugates.
Machulkin AE, Skvortsov DA, Ivanenkov YA, Ber AP, Kavalchuk MV, Aladinskaya AV, Uspenskaya AA, Shafikov RR, Plotnikova EA, Yakubovskaya RI, Nimenko EA, Zyk NU, Beloglazkina EK, Zyk NV, Koteliansky VE, Majouga AG. Machulkin AE, et al. Among authors: shafikov rr. Bioorg Med Chem Lett. 2019 Aug 15;29(16):2229-2235. doi: 10.1016/j.bmcl.2019.06.035. Epub 2019 Jun 20. Bioorg Med Chem Lett. 2019. PMID: 31248772
Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom.
Zyk NY, Ber AP, Nimenko EA, Shafikov RR, Evteev SA, Petrov SA, Uspenskaya AA, Dashkova NS, Ivanenkov YA, Skvortsov DA, Beloglazkina EK, Majouga AG, Machulkin AE. Zyk NY, et al. Among authors: shafikov rr. Bioorg Med Chem Lett. 2022 Sep 1;71:128840. doi: 10.1016/j.bmcl.2022.128840. Epub 2022 May 31. Bioorg Med Chem Lett. 2022. PMID: 35661685
12 results